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  Bulking Steroids:

  Anabol 5mg British Dispensary
Anabol 50mg - British Dragon
Anabol 50mg, C&K, China
Anabol 5mg - C&K
Anadrol 50 / oxymetholone
Anapolon 50 mg
Anavar
Andriol / Testosterone Undecanoate
ANDRIOL TESTOCAPS 40mg
Androlic 50mg British Dragon
Androlic 50mg British Dispensary
Androlic 50mg, C&K, China
Averbol 25
BONALONE (Oxymetholone)
Clomid 50mg, Global Napi
Cypioject 10 ml vial (200 mg/ml) Testosterone cypionate
Cypionax (Testosterone cypionate)
Danabol, 10mg, 500tabs, DS
Deca Durabolin (Norma)
Deca Durabolin (Organon)
Deca-durabolin 100mg
Deca-durabolin 50mg
Decabol 250 British Dragon
Decadubol-100
Decaject 200
Dubol-100
Dubol-50
Durabol British Dragon
Durabol 200
Durabolin 25
Halotestex British Dragon
Halotestin 5mg
Mastabol 100 British Dragon
Mastabol Depot 200 BD
Metanabol 5mg Poland, Jelfa
Methanabol 10mg 100tabs British Dragon
Methanabol 10mg 500tabs BD
Methanabol 50mg 100tabs BD
Methandriol Dipropionate 75
Methandrostenoloni - 5mg
Nandrolone decanoate
Nandrolone Phenylpropionate
Naposim 5mg
Omnadren
Oxanabol 10mg 50tabs
Oxanabol, 5mg, C&K
Oxydrol 50Mg, 100tabs BritishDragon
Primoteston Depot 1ml amp
Restandol
SustaJect 250 (Ec labs - Eurochem)
Sustanon 250 Pakistan
Sustanon 250mg/1ml Nile
Testabol Cypionate
Testabol Depot, British Dragon
Testabol Enanthate British Dragon
Testabol Propionate 100, 10ml
Testen-250
TESTENON
Testex Elmu Prolongatum 250mg/2ml
TestoJect / 4x testosterone blend
Testosteron Depo 1ml/amp
Testosterone cypionate 200mg
Testosterone Enanthate 250
Testosterone Enanthate 250 Norma
Testosterone Propionate 50mg/ml, Farmak
Testosterone suspension / Aquaviron
Testoviron Depot / Schering
TESTOVIS / testosterone-propionate
Trenabol 75 / British Dragon
Tri-Trenabol 150 BD
Turanabol 10mg

  Cutting Steroids:

  Anadiol Depot, Ilium
Boldabol / British Dragon
Bonavar / Oxandrolone
Cetabon (anabolic formula)
Danabolan
Equipoise 50mL / 50mL - 50mg/1ml
Fluoxymesterone 10mg
Stanabolic 50mg/ml Ilium
Lasix (furosemide)
Orabolin / etylestrenol, 2 mg/tab
PARATABS - Parabolan (trenbolone acetate), 60 tabs (25 mg/tab)
Primobol 100 British Dragon
Primobol tabs, British Dragon
Primobolan Depot
Primoject 10ml
Stanabol 10mg
Stanabol 50injectable (Stanozolol)
Stanabol 50mg British Dragon
Stanabol 50mg C&K
Stanabol 5mg, C&K
Stanoject / Stanozolol
STANOL (stanozolol) 5 mg 200tab
Stanol 50mg/1ml
Stanol 50mg/1ml
STANOZOLOL 1ml x 50mg/ml, LA
Stanozolol 10mg 100Tabs / LA, Italy
STANOZOLOL 50mg/ml ( ILIUM )
Testolic 2ml testosteron propianate
TESTOPIN-100 2 ml vial
Trenabol depot 100mg/1ml
Trenbolone Acetate tabs, BD
Virormone 2ml (Testosterone Propionate) 100mg/1ml
Voltaren 75

  Man's Health:

  Caverject 10mcg, Syringes
Caverject 20mcg
Caverject 20mcg
Propecia 1mg (Finasteride) 28 tabs
Viagra

  Human Hormones:

  Choriomon
Choriomon 15000IU
Igtropin IGF1 LR3 100mcg
Jintropin 10IU(100IU/box)
Jintropin 10IU(200IU/kit)
Jintropin 4IU(40IU/box)
Jintropin 4IU(80IU/box)
Pregnyl 5000 IU Organon
Pregnyl 3 X 5000 IU (HCG)

  Anti Estrogens:

  Anastrozole, - British Dragon
Arimidex / Anastrozole
Aromasin 20 mg / British Dragon
Aromasin 25 mg / Pfizer
Aromasin 25 mg
Clenbuterol / Hubei Huangshi
Clomid 50mg C&K
Clomid 50mg, Aventis
Clomid 50mg, Brunno Farmaceutici
Clomifen 25 mg
Clomiphene 50mg
Clomiphene citrate 50mg
Mesterolone BD (Proviron)
Nolvadex 10mg
Nolvadex, 20mg, AstraZeneca
Nolvadex, 40mg, AstraZeneca
Nolvadex, 50mg, C&K China
Omifin 50 mg 30 tabs
Proviron 25mg (Mesterolone)
Provironum 25mg Schering
Tamoxifen 20mg British Dragon
Teslac (Testolactone) 50mg / 100 tabs

  Anti Depressants:

  ADDERALL XR 15MG CAPSULES
Dumirox (Fluvoxamine) 50mg
Rivotril (CLONAZEPAM) 0.5 mg
Rivotril (CLONAZEPAM) 2 mg
Rivotril (CLONAZEPAM) 2 mg
Rohypnol (Flunitrazepam) 1mg
Valium (DIAZEPAM) 10mg
Valium (DIAZEPAM) 5mg

  Head Ache:

  Maxalt (Rizatripan) 10 mg
Relpax 40mg
Zomigon (Zolmitriptane) 2.5mg

  Herpes:

  Famvir (Famciclovir) 125 mg
Viranet (Valacyclovir) 500mg
Zovirax (Acyclovir) 15 gr

  Muscle Relaxers:

  Baclofen 25mg
Muscoril Caps 20 x 4 mg
Norgesic (Orphenadrine)

  Pain Releaf:

  Advil (Ibuprofen) 200mg
Celebrex 200mg
Mesulid (Nimesulide) 100mg
Movatec (Meloxicam) 15mg
Naprosyn 500mg
Oruvail (Ketoprofen) 200mg
Vioxx 25mg

  Quit Smoking:

  Zyban (bupropion) 150 mg

  Skin Care:

  Harifin 5 (Finasteride) 5mg

  Weight Loss:

  Cynomel 0,025mg (25mcg) (Cytomel / T3) / Liothyronine Sodium
Cytomel / T4 50 mg
Phentermine (blue/clear) 30mg. 100 Caps
Reducil 28tabs 15mg
TRIACANA 0.35 mcg

  Anxiety:

  Vespar

  Genital Warts:

  Aldara cream 5% (Imiquimod)
Wartek (Podophyllotoxin) cream

Aromasin 20mg / Exemestane Tablets / British Dragon


Name Manufacturer Volume Price $ Price Quantity
Aromasin 20mg / Exemestane Tablets / NEWBritish Dragon, Thailand50 tabs $130  €118  /

 
Aromasin 20mg / Exemestane Tablets / British Dragon
 
Aromasin 20mg / Exemestane Tablets / British Dragon
Generic name: Exemestane

by Anthony Roberts -- Aromasin (Exemestane) is one of those weird compounds that nobody really knows what to do with. What we generally hear about it makes it very uninteresting…It’s a third generation Aromatase Inhibitor (AI) just like Arimidex (Anastrozole) and Femera (Letrozole). Both of those two drugs are very efficient at stopping the conversion of androgens into estrogen, and since we have them, why bother with Aromasin? It’s a little harder to get than the other two commonly used aromatase inhibitors, because it’s not in high demand, and there’s never been a readily apparent advantage to using it. And I mean…lets face it: It’s awkward-sounding. Aromasin doesn’t have much of a ring to it, and exemestane is even worse. Arimidex has a bunch of cool abbreviations ("A-dex" or just ‘dex) and even Letrozole is just "Letro" to most people. Where’s the cool nickname for Aromasin/exemestane? A-Sin? E-Stane? It just doesn’t work. It’s the black sheep of AIs. And why do we even need it when we have Letrozole, which is by far the most efficient AI for stopping aromatization (the process by which your body converts testosterone into estrogen)? Letro can reduce estrogen levels by 98% or greater; clinically a dose as low as 100mcgs has been shown to provide maximum aromatase inhibition (2)! So why would we need any other AIs? Well, first of all, estrogen is necessary for healthy joints (3) as well as a healthy immune system (4). So getting rid of 98% of the estrogen in your body for an extended period of time may not be the best of ideas. This may be useful on an extreme cutting cycle, leading up to a bodybuilding contest, or if you are particularly prone to gyno, but certainly can’t be used safely for extended periods of time without compromising your joints and immune system.

So that leaves us with Arimidex, which isn’t as potent as Letrozole, but at . 5mgs/day will still get rid of around half (50%) of the estrogen in your body. Problem solved, right? Use Arimidex on your typical cycles, and if you are very prone to gyno or are getting ready for a contest, use Letro.

But what about Post Cycle Therapy (PCT)?

I think at this point most people are sold on the use of Nolvadex (Tamoxifen Citrate) instead of Clomid for PCT, since both compete estrogen at the receptor site, both increase serum test levels, and both drugs may also alter blood lipid profiles favorably (6). But since 20mgs of Tamoxifen is equal to 150mgs of clomid for purposes of testosterone elevation, FSH and LH, but Tamoxifen doesn’t decrease the LH response to LHRH (6) I think most people agree to Nolvadex’s superiority for PCT.

I’ve always been in favor of using Nolvadex during PCT, along with an AI, because reducing estrogen levels has been positively correlated with an increase in testosterone (7) so in my mind, it’s be beneficial to increase testosterone by as many mechanisms as possible while trying to recover your endogenous testosterone levels after a cycle. SO which AI do we use? Letro or A-dex? Well, why don’t we just keep using whichever one we used during the cycle, and add in some Nolvadex? Unfortunately, Nolvadex will significantly reduce the blood plasma levels of both Letrozole as well as Arimidex (8). So if we choose to use one of them with our Nolvadex on PCT, we’re throwing away a bit of money as the Nolvadex will be reducing their effectiveness.

This, of course, is where Aromasin comes in, at 20-25mgs/day.

Aromasin, at that dose, will raise your testosterone levels by about 60%, and also help out your free to bound testosterone ratio by lowering levels of Sex Hormone Binding Globulin (SHBG), by about 20% (12)…SHBG is that nasty enzyme that binds to testosterone and renders it useless for building muscle. But what about using it along with Nolvadex for PCT?

To understand why Aromasin may be useful in conjunction with Nolvadex while both Letro and A-dex suffer reduced effectiveness, we’ll need to first understand the differences between a Type-I and Type-II Aromatase Inhibitor. Type I inhibitors (like Aromasin) are actually steroidal compounds, while typeII inhibitors (like Letro and A-dex) are non-steroidal drugs. Hence, androgenic side effects are very possible with Type-I AIs, and they should probably be avoided by women. Of course, there are some similarities between the two types of AIs…both type I & type II AIs mimic normalsubstrates (essentially androgens), allowing them to compete with the substrate for accessto the binding site on the aromatase enzyme. After this binding, thenext step is where things differ greatly for the two different types of AI’s. In the case of a type-I AI, the noncompetitive inhibitorwill bind, and the enzyme initiates a sequence of hydroxylation; this hydroxylation produces an unbreakable covalent bond betweenthe inhibitor and the enzyme protein. Now, enzyme activity is permanently blocked; even if all unattached inhibitor is removed. Aromatase enzyme activity can only be restored by new enzyme synthesis. Now, on the other hand, competitive inhibitors, called type II AI’s, reversibly bind to the active enzymesite, and one of two things can happen: 1. ) either no enzyme activity is triggered or 2. ) the enzyme is somehow triggered withouteffect. The type II inhibitor can now actually disassociate from the binding site, eventually allowing renewed competition between the inhibitor and the substratefor binding to the site. This means that the effectiveness of competitive aromatase inhibitors depends on the relative concentrations and affinitiesof both the inhibitor and the substrate, while this is not so for noncompetitive inhibitors. Aromasin is a type-I inhibitor, meaning that once it has done its job, and deactivated the aromatase enzyme, we don’t need it anymore. Letrozole and Arimidex actually need to remain present to continue their effects. This is possibly why Nolvadex does not alter the pharmacokinetics of Aromasin (11).

Before we close the book on Aromasin, it’s worth noting that you can (and should) still use one of the non-steroidal AIs during your cycle to reduce estrogen, if necessary. When you are ready for PCT, you can then switch over to Aromasin and still experience the full effects of an AI, since there is no cross-over tolerance experienced between steroidal and non-steroidal AIs (9). Since Aromasin is about 65% efficient at suppressing estrogen (10), it’s certainly a very powerful agent, especially considering you won’t experience reduced effectiveness because of your concurrent use of Nolvadex or from any sort of tolerance developed by using other AIs on your cycle(9). There is also a decent amount of preclinical data suggesting that Aromasin has a beneficial effect on bone mineral metabolism that isnot seen with non-steroidal agents, and it may also have beneficial effects on lipid metabolism that are notfound in the non-steroidal Letro and A-dex (9).

Finally, as we’re going to be using Nolvadex for PCT anyway, and we ought to be using an AI with it for maximum recovery…I think Aromasin- considering it’s compatibility with Nolvadex and beneficial effects on bone mineral content and lipid profile, has finally stopped being the black sheep of AIs and found a home in our Cycles.








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